ActiTide™ NP1 / Nonapeptide-1

Nkọwa dị mkpirikpi:

Alfa-Melanocyte-Stimulating Hormone (α-MSH), peptide 13-amino acid, na-ejikọta ya na onye na-anabata ya (MC1R) iji mee ka ụzọ melanin rụọ ọrụ, na-eme ka mmepụta melanin dịkwuo elu na akpụkpọ ahụ gbara ọchịchịrị. ActiTide ™ NP1, peptide biomimetic emebere iji ṅomie usoro nke α-MSH, na-egbochi ike njide α-MSH na onye nata ya. Site na igbochi ịgbalite ụzọ melanin na isi mmalite ya, ActiTide ™ NP1 na-ebelata njikọ nke melanin ma gosipụta nrụpụta akpụkpọ ahụ.


Nkọwa ngwaahịa

Mkpado ngwaahịa

Aha ika ActiTide™ NP1
CAS Mba. /
Aha INCI Nonapeptide-1
Ngwa Usoro nkpuchi, usoro ude, usoro serum
ngwugwu 100g / karama, 1kg / akpa
Ọdịdị Na-acha ọcha na-acha ọcha ntụ ntụ
Peptide ọdịnaya 80.0 min
Solubility Soluble na mmiri
Ọrụ Usoro Peptide
Ndụ nchekwa Afọ 2
Nchekwa Ekwesịrị ịchekwa ya na 2 ~ 8 Celsius C n'ime akpa mechiri emechi
Usoro onunu ogwu 0.005% -0.05%

Ngwa

 

Isi ọnọdụ

ActiTide ™ NP1 bụ ihe na-acha ọcha dị ike nke na-elekwasị anya na mbido mbụ nke usoro ịgba ọchịchịrị. Site na itinye aka na mmepụta melanin na isi iyi ya, ọ na-enye njikwa ụda akpụkpọ ahụ dị elu ma na-ebelata ọdịdị nke ntụpọ aja aja.

Isi Mechanism nke Action

1. Ntinye aka isi mmalite:Na-egbochi mgbaàmà mgbake Melanogenesis na-egbochi njikọ α-melanocyte-stimulating hormone (α-MSH) na onye na-anabata MC1R na melanocytes.
Nke a na-ekewa ozugbo "mgbama mmalite" maka mmepụta melanin, na-akwụsị usoro njikọ na-esote na isi iyi ya.
2. Mgbochi usoro:Na-egbochi ịgbalite Tyrosinase Ọzọkwa na-egbochi ịgbalite tyrosinase, enzyme bụ isi dị mkpa maka njikọ melanin.
Omume a na-egbochi usoro melanogenesis nke ọma iji lụso ọzịza anụ ahụ ọgụ nke ọma ma gbochie ịmepụta ntụpọ aja aja.
3. Njikwa mmepụta: Na-egbochi mmepụta Melanin karịrị akarị Site na usoro abụọ dị n'elu.
N'ikpeazụ, ọ na-eme ka njikwa nke ọma na "mpụta oke" nke melanin, na-egbochi ụda akpụkpọ ahụ na-adịghị mma na ịba ụba nke hyperpigmentation.

Ntuziaka mgbakwunye nhazi

Iji chekwaa ọrụ nke ngwa ahụ ma zere ikpughe ogologo oge na oke okpomọkụ, a na-atụ aro ka ịgbakwunye ActiTide ™ NP1 n'oge ikpeazụ jụrụ oyi nke nhazi. Okpomọkụ sistemu kwesịrị ịdị n'okpuru 40 Celsius C n'oge ntinye.

Ngwa ngwaahịa akwadoro

Ngwa a dabara adaba maka usoro ịchọ mma dị iche iche na-arụ ọrụ, gụnyere:
1. Akpụkpọ anụ na-egbuke egbuke & ngwaahịa na-egbuke egbuke
2. Na-acha ọcha / na-amụba ọbara ọbara na ude
3. mgbochi-ọchịchịrị ntụpọ na hyperpigmentation ọgwụgwọ

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